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EUROPEAN PATENTS AND PATENT APPLICATIONS

H.F. DeLuca, L. A. Plum, R. R. SiciÅ„ski, I. Sibilska. 3-Desoxy-2-methylene-19-nor-vitamin D analogs and their uses. EP2721004 B1 (26 July 2017)

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H. F. DeLuca, L. A. Plum, I. Sibilska, R. R. Siciński. 3-Desoxy-2-methylene-19-nor-vitamin D analogs and their uses. EP 2768804 A1 (27 Aug 2014).

 

H. F. DeLuca, L. A. Plum, I. Sibilska, R. R. Siciński. 3-Desoxy-2-methylene-19-nor-vitamin D analogs and their uses. EP 2768803 A1 (27 Aug 2014).

 

M. Clagett-Dame, H. F. DeLuca, L. A. Plum, I. Sibilska, R. R. Siciński. 3-Desoxy-2-methylene-19-nor-vitamin D analogs and their uses. EP 2721004 A1 (23 Apr 2014).

 

K. M. Barycka, R. Barycki, M. Clagett-Dame, H. F. DeLuca, K. Płonska-Ocypa, L. A. Plum, I. Sibilska, R. R. Siciński. 1-Desoxy-2-methylene-19-nor-vitamin D analogs and their uses. EP 2483240 A2 (08 Aug 2012).

 

H. F. DeLuca, M. Clagett-Dame, P. Grzywacz, N. J. Nieves, K. PÅ‚oÅ„ska-Ocypa, L. A. Plum, R. R. SiciÅ„ski. 13,13-Dimethyl-des-C,D analogs of 1α,25-dihydroxy-19-nor-vitamin D3 compounds and topical composition dosage forms and methods of treating skin conditions thereof. EP 2247563 A1 (10 Nov 2010).

 

H. F. DeLuca, M. Clagett-Dame, A. Głębocka, L. A. Plum, R. R. Siciński. 2-Methylene-20-methyl-19,24,25,26,27-pentanor-vitamin D analogs. EP 2240438 A1 (20 Oct 2010).

 

H. F. DeLuca, M. Clagett-Dame, A. GÅ‚Ä™bocka, L. A. Plum, R. R. SiciÅ„ski. 1α-Hydroxy-2-(3'-hydroxypropylidene)-19-nor-vitamin D compounds and methods of making and use thereof. EP 2010483A2 (7 Jan 2009). 

 

H. F. DeLuca, A. GÅ‚Ä™bocka, R. R. SiciÅ„ski, L. A. Plum, M. Clagett-Dame. 1α-Hydroxy-2-(3'-hydroxypropylidene)-19-nor-vitamin D compounds with a 1,1-dimethylpropyl side chain. EP 2004597A2 (24 Dec 2008). 

 

H. F. DeLuca, R. R. Siciński, A. Głębocka, L. A. Plum, M. Clagett-Dame. 19-Nor-vitamin D analogs with 1,2, or 3,2 heterocyclic ring. EP 2001860A2 (17 Dec 2008).

 

H. F. DeLuca, R. R. SiciÅ„ski, P. K. Grzywacz, (20S)-1α-Hydroxy-2 -methyl and 2α-methyl-19-nor-vitamin D3 and their uses. EP 1496914B1 (26 Nov 2008).

 

H. F. DeLuca, R. R. Siciński. 2-Ethyl and 2-ethylidene-19-nor-vitamin D compounds. EP 1286962B1 (25 Jun 2008).

 

H. F. DeLuca, K. PloÅ„ska-Ocypa, R. R. SiciÅ„ski, P. Grzywacz, L. A. Plum, M. Clagett-Dame. Des-C,D analogs of 1α,25-dihydroxy-19-norvitamin D3. EP 1931324A2 (18 Jun 2008).

 

H. F. DeLuca, P. K. Grzywacz, R. R. Siciński. Synthesis of indole thiazole compounds as ligands for the AH receptor. EP 1480951B1 (7 May 2008).

 

H. F. DeLuca, R. R. SiciÅ„ski, L. A. Plum, M. Clagett-Dame. 2 -Methyl-19-nor-(20S)-1α-hydroxy-bishomopregnacalciferol and its uses. EP 1846369A2 (24 Oct 2007).

 

H. F. DeLuca, R. R. SiciÅ„ski, L. A. Plum, M. Clagett-Dame, S. Gowlugari. 2α-Methyl-19-nor-1α-hydroxy-homopregnacalciferol and its uses. EP 1838667A2 (3 Oct 2007).

 

H. F. DeLuca, R. R. Siciński, S. Gowlugari, L. A. Plum, M. Clagett-Dame, 2-Alkylidene-19-nor-vitamin D compounds and their therapeutic uses. EP 1268416B1 (26 Sept 2007).

 

H. F. DeLuca, R. Barycki, P. K. Grzywacz, L. A. Plum, R. R. Siciński. 2-Alkylidene-18,19-dinor-vitamin D compounds. EP 1735277A1 (27 Dec 2006).

 

H. F. DeLuca, S. Gowlugari, R. R. SiciÅ„ski. Method of synthesizing 1α-hydroxy-2-methylene-19-nor-homopregnacalciferol. EP 1490332B1 (29 Nov 2006).

 

H. F. DeLuca, R. R. SiciÅ„ski, S. Gowlugari, L. A. Plum, M. Clagett-Dame, 1α-Hydroxy-2-methylene-19-nor-homopregnacalciferol and its therapeutic applications. EP 1315504B1 (18 Aug 2004).

 

H. F. DeLuca, R. R. Siciński. 2-Alkyl-19-nor-vitamin D compounds, EP 0971888B1 (29 Oct 2003).

 

H. F. DeLuca, H. K. Schnoes, R. R. Siciński, X. Jia. All-trans retinol metabolite. EP 1012149B1 (25 Sept 2002).

 

H. F. DeLuca, R. R. SiciÅ„ski. 2-Alkylidene-19-nor-vitamin D compounds. EP 0970047B1 (9 Nov 2002). 

 

H. F. DeLuca, R. R. SiciÅ„ski, K. L. Perlman. 18,19-Dinor-vitamin D compounds. EP 793649B1 (03 Feb 1999). 

 

H. F. DeLuca, R. R. SiciÅ„ski. (E)-20(22)-Dehydrovitamin D compounds. EP 726892B1 (30 Dec 1998). 

 

H. F. DeLuca, R. R. SiciÅ„ski. Iodo vitamin D3 compounds and method for preparing same. EP 0624573B1 (15 Oct 1997). 

 

H. F. DeLuca, K. L. Perlman, R. R. SiciÅ„ski. 19-Nor-vitamin D3 compounds with substituent at 2-position. EP 0619306B1 (11 Sept 1996). 

 

H. F. DeLuca, H. K. Schnoes, K. L. Perlman, R. R. SiciÅ„ski, J. M. Prahl. 19-Nor-vitamin D compounds. EP 387077B1 (19 Jan 1994). 

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